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You are here:Home-Inhibitors & Agonists-GPCR-Chemokine Receptor (CCR and CXCR)

Request The Product List ofChemokine Receptor (CCR and CXCR) Chemokine Receptor (CCR and CXCR)

Cat. No. Product Name CAS No. Information
H9623

CCR2 Inhibitor SD-24

 		1237502-86-1

CCR2 inhibitor SD-24 is a potent selective CCR2 antagonist with pKi of 8.5.
H9615

CCR4-351

 		2206788-99-8

CCR4-351 is a potent, selective, orally bioavailable CCR4 antagonist with IC50 of 40 nM ;CCR4-IN-31 exhibited high potency in distinct functional assays in addition to good in vitro and in vivo ADME properties.CCR4-IN-31 potentiate antitumor immune responses.
H9132

Cenicriviroc Mesylate

 		497223-28-6

Cenicriviroc Mesylate (TAK-652 Mesylate) is a dual CCR2/CCR5 antagonist, also inhibits both HIV-1 and HIV-2, and displays potent anti-inflammatory and antiinfective activity.
H9131

Cenicriviroc

 		497223-25-3

Cenicriviroc (TAK-652) is an orally active, dual CCR2/CCR5 antagonist, also inhibits both HIV-1 and HIV-2, and displays potent anti-inflammatory and antiinfective activity.
H9065

ACT-1004-1239

 		2178049-58-4

ACT-1004-1239 is a potent, selective, orally available CXCR7 antagonist with IC50 value of 3.2 nM ,Oral administration of ACT-1004-1239 in mice up to 100 mg/kg led to a dose-dependent increase of plasma CXCL12 concentration.
H8993

KAND 567

 		911715-90-7

AZD8797 is an allosteric non-competitive and orally active antagonist of the human CX3CR1 receptor; antagonizes CX3CR1 and CXCR2 with Kis of 3.9 and 2800 nM, respectively.
H8849

Lazucirnon

 		1251528-23-0

Lazucirnon is a potent Pharmaceutical formulations CCR3 antagonists.
H3215

α-NETA

 		31059-54-8

A small molecule CMKLR1 antagonist that inhibits chemerin-stimulated β-arrestin2 association with CMKLR1 (EC50=9.7 nM); inhibits chemerin-triggered CMKLR1+ cell migration, suppresses CNS autoimmune inflammatory disease in vivo; also inhibits choline acetyltransferase with IC50 of 9 uM.
H3214

VUF11403

 		1378524-61-8

A potent CXCR7 (ACKR3) agonist.
H3213

VUF11207 fumarate

 		1378524-41-4

A potent CXCR7 (ACKR3) agonist with EC50 of 1.6 nM; inducse recruitment of β-arrestin2 and subsequent internalization of CXCR7 in cells.

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