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You are here:Home-Inhibitors & Agonists-Nuclear Receptor/Transcription Factor-Rev-ErbA

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Cat. No. Product Name CAS No. Information
H5957

SR 8278

 		1254944-66-5

SR 8278 is the first synthetic antagonist of the nuclear heme receptor Rev-ErbA, inhibits the REV-ERBα transcriptional repression activity with EC50 of 0.47 uM in HEK293 cells.
H5956

GSK-2945

 		1438071-12-5

GSK-2945 is a potent and selective small molecule Rev-Erbα agonist with EC50 of 50 nM, displays >1,000-fold selectivity over LXRα; inhibits LPS induction of IL-6 production and to upregulate expression of ABCA1 in human THP-1 cells; demonstrates in vivo bioavailability and orally active.

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